SCHEMBL7424358

SCHEMBL7424358

CC(C)CC(NCC(C(=O)O)c1ccc(-c2ccc(C(F)(F)F)cc2)o1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.49
PSEN2 P49810 1/20 0.49
APH1B Q8WW43 1/20 0.49
NCSTN Q92542 1/20 0.49
APH1A Q96BI3 1/20 0.49
PSENEN Q9NZ42 1/20 0.49
TP53 P04637 1/20 0.40
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
APP P05067 1/20 0.37
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MMP13 P45452 2/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416089 0.87 ALOX5 (0.44) SORT1ERCC5FEN1ALOX5
SCHEMBL7420893 0.86 ALDH1A1 (0.41) CYP1A2CYP2C19ALDH1A1MMP13MMP1
SCHEMBL7421514 0.85 ALDH1A1 (0.44) ALDH1A1SORT1ERCC5FEN1GRN
SCHEMBL7419841 0.83 KDM4E (0.44) ALDH1A1MMP13
SCHEMBL7418370 0.83 PSEN1 (0.60) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7427850 0.82 SORT1 (0.39) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7418844 0.81 SORT1 (0.41) AKR1C3AKR1C2CYP2C19ALDH1A1SORT1
SCHEMBL7427316 0.80 SORT1 (0.46) CYP2C19ALDH1A1SORT1GRNACE
SCHEMBL7421684 0.79 S1PR4 (0.40) CYP2C19ALDH1A1MMP13MMP1MMP2
SCHEMBL7425626 0.78 MAPK1 (0.47) ALDH1A1SORT1GRN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed