SCHEMBL7426929

SCHEMBL7426929

NC(=O)c1ccc2c(c1)N(C(=O)Cc1cccnc1)CC2.NCc1cccc(N(CC(=O)O)C(=O)c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
ROCK1 Q13464 2/20 0.38
EIF2AK3 Q9NZJ5 2/20 0.38
LCK P06239 1/20 0.38
AURKB Q96GD4 1/20 0.38
EIF2AK1 Q9BQI3 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
STAT3 P40763 1/20 0.37
RIPK1 Q13546 2/20 0.37
NPY2R P49146 1/20 0.37
TNKS O95271 1/20 0.35
PARP1 P09874 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
PARP4 Q9UKK3 1/20 0.35
PARP3 Q9Y6F1 1/20 0.35
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7427969 0.93 ALDH1A1 (0.46) CYP11B1CYP11B2ALDH1A1MAPTROCK1
Trifluoroacetic Acid SCHEMBL5213690 0.91 CYP11B1 (0.41) CYP11B1CYP11B2ALDH1A1MAPTROCK1
SCHEMBL7428011 0.90 ALDH1A1 (0.39) CYP11B1CYP11B2ALDH1A1MAPTROCK1
Trifluoroacetic Acid SCHEMBL7433118 0.89 RIPK1 (0.39) CYP11B1CYP11B2ALDH1A1ROCK1EIF2AK3
SCHEMBL7434744 0.86 OPRD1 (0.36) ALDH1A1MAPTROCK1TSHRRIPK1
SCHEMBL7424730 0.85 ROCK1 (0.37) CYP11B1CYP11B2ALDH1A1ROCK1EIF2AK3
Trifluoroacetic Acid SCHEMBL5210778 0.84 RIPK1 (0.39) CYP11B1CYP11B2ALDH1A1ROCK1EIF2AK3
Hydrochloric Acid SCHEMBL5244756 0.84 ALDH1A1 (0.39) CYP11B1CYP11B2ALDH1A1MAPTROCK1
Trifluoroacetic Acid SCHEMBL5208180 0.84 RIPK1 (0.42) CYP11B1CYP11B2ALDH1A1MAPTROCK1
Trifluoroacetic Acid SCHEMBL5210860 0.83 RIPK1 (0.42) CYP11B1CYP11B2ALDH1A1MAPTROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192135-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2002-04-03 EP disclosed
WO-2000076970-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2000-12-21 WO disclosed