SCHEMBL7424730

SCHEMBL7424730

NC(=O)c1ccc2c(c1)N(C(=O)Cc1c[nH]cn1)CC2.NCc1cccc(N(CC(=O)O)C(=O)c2ccccc2)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.37
ALDH1A1 P00352 1/20 0.35
RIPK1 Q13546 1/20 0.34
PTGIR P43119 1/20 0.33
OPRM1 P35372 3/20 0.33
OPRD1 P41143 3/20 0.33
OPRK1 P41145 2/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
F2 P00734 2/20 0.32
EIF2AK1 Q9BQI3 1/20 0.32
EIF2AK3 Q9NZJ5 1/20 0.32
XIAP P98170 1/20 0.32
BIRC2 Q13490 1/20 0.32
ADAMTS4 O75173 1/20 0.31
ROCK2 O75116 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5213379 0.92 RIPK1 (0.36) ROCK1ALDH1A1RIPK1OPRM1OPRD1
SCHEMBL7427969 0.89 ALDH1A1 (0.46) ROCK1ALDH1A1RIPK1OPRM1OPRD1
SCHEMBL7428011 0.87 ALDH1A1 (0.39) ROCK1ALDH1A1RIPK1OPRM1OPRD1
SCHEMBL7426929 0.85 CYP11B1 (0.45) ROCK1ALDH1A1RIPK1OPRM1OPRD1
SCHEMBL7434744 0.83 OPRD1 (0.36) ROCK1ALDH1A1RIPK1OPRM1OPRD1
Trifluoroacetic Acid SCHEMBL7433118 0.82 RIPK1 (0.39) ROCK1ALDH1A1RIPK1CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL5244756 0.81 ALDH1A1 (0.39) ROCK1ALDH1A1RIPK1OPRM1OPRD1
Hydrochloric Acid SCHEMBL5212001 0.80 EIF2AK3 (0.37) ROCK1ALDH1A1RIPK1CYP11B1CYP11B2
Trifluoroacetic Acid SCHEMBL5208180 0.80 RIPK1 (0.42) ROCK1ALDH1A1RIPK1CYP11B1CYP11B2
Trifluoroacetic Acid SCHEMBL8041708 0.80 RIPK1 (0.37) ROCK1ALDH1A1RIPK1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192135-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2002-04-03 EP disclosed
WO-2000076970-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2000-12-21 WO disclosed