Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL7433118

NC(=O)c1ccc2c(c1)N(C(=O)Cc1ccncc1)CC2.NCc1cccc(N(CC(=O)O)C(=O)c2ccccc2)c1.O=C(O)C(F)(F)F.O=C(O)C(F)(F)F

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ALDH1A1 P00352 1/20 0.38
ROCK1 Q13464 5/20 0.38
EIF2AK3 Q9NZJ5 3/20 0.35
ACHE P22303 1/20 0.35
ROCK2 O75116 2/20 0.35
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
EIF2AK1 Q9BQI3 2/20 0.33
LCK P06239 1/20 0.33
AURKB Q96GD4 1/20 0.33
NPY2R P49146 1/20 0.33
F2 P00734 2/20 0.33
F10 P00742 2/20 0.33
TPSAB1 Q15661 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5210778 0.96 RIPK1 (0.39) RIPK1CYP11B1CYP11B2ALDH1A1ROCK1
Trifluoroacetic Acid SCHEMBL5208180 0.91 RIPK1 (0.42) RIPK1CYP11B1CYP11B2ALDH1A1ROCK1
SCHEMBL7427969 0.91 ALDH1A1 (0.46) RIPK1CYP11B1CYP11B2ALDH1A1ROCK1
Trifluoroacetic Acid SCHEMBL5210860 0.90 RIPK1 (0.42) RIPK1CYP11B1CYP11B2ALDH1A1ROCK1
Trifluoroacetic Acid SCHEMBL5213690 0.89 CYP11B1 (0.41) RIPK1CYP11B1CYP11B2ALDH1A1ROCK1
SCHEMBL7426929 0.89 CYP11B1 (0.45) RIPK1CYP11B1CYP11B2ALDH1A1ROCK1
Trifluoroacetic Acid SCHEMBL8041708 0.88 RIPK1 (0.37) RIPK1ALDH1A1ROCK1TPSAB1
Trifluoroacetic Acid SCHEMBL7430442 0.87 RIPK1 (0.38) RIPK1ALDH1A1ROCK1F2F10
Trifluoroacetic Acid SCHEMBL7432346 0.87 RIPK1 (0.37) RIPK1ALDH1A1ROCK1ACHENPY2R
Trifluoroacetic Acid SCHEMBL5212450 0.87 RIPK1 (0.39) RIPK1ALDH1A1ROCK1ACHENPY2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192135-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2002-04-03 EP disclosed
WO-2000076970-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2000-12-21 WO disclosed