SCHEMBL7427872

SCHEMBL7427872

CCOC(=O)c1ccc2c(cnn2CC(=O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.48
EGFR P00533 1/20 0.46
ERBB2 P04626 1/20 0.46
PLA2G4A P47712 1/20 0.46
HSD17B10 Q99714 2/20 0.46
POLB P06746 1/20 0.46
TSHR P16473 1/20 0.46
SIRT2 Q8IXJ6 2/20 0.45
SIRT1 Q96EB6 2/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
RAB9A P51151 4/20 0.44
NPC1 O15118 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 2/20 0.44
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL904672 0.88 MAPT (0.48) EGFRERBB2SIRT2SIRT1CA12
SCHEMBL7426302 0.88 EGFR (0.45) EGFRERBB2PLA2G4AHSD17B10POLB
SCHEMBL7425784 0.88 KMO (0.60) KMOEGFRERBB2SIRT2SIRT1
SCHEMBL7428104 0.86 PLA2G4A (0.46) EGFRERBB2PLA2G4AHSD17B10POLB
SCHEMBL7425711 0.84 POLB (0.42) EGFRERBB2PLA2G4AHSD17B10POLB
SCHEMBL4957912 0.84 HTR2A (0.46) KMOEGFRERBB2TSHRSIRT2
SCHEMBL4959328 0.82 MAOA (0.43) KMOEGFRERBB2TSHRSIRT2
SCHEMBL8684617 0.81 MAOA (0.43) KMOEGFRERBB2PLA2G4ATSHR
SCHEMBL3436319 0.81 CCNC (0.49) HSD17B10SIRT2SIRT1CA12CA1
Hydrochloric Acid SCHEMBL8683583 0.81 MAOA (0.42) KMOEGFRERBB2PLA2G4ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6489333-B2 HETEROCYCLIC COMPOUNDS CONTAINING A GUANIDINE MIMIC, FOR INHIBITION OF CELL ADHESION, TREATMENT OF ANGIOGENESIS DISORDERS, INFLAMMATION, CANCER METASTASIS, DIABETIC RETINOPATHY, THROMBOSIS, RESTENOSIS, MACULAR DEGENERATION BRISTOL - MEYERS SQUIBB PHARMA COMPANY 2002-12-03 US disclosed
US-20010044535-A1 Integrin antagonists BRISTOL-MYERS SQUIBB PHARMA COMPANY 2001-11-22 US disclosed
EP-1054871-A2 PYRIMIDINES AND TRIAZINES AS INTEGRIN ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2000-11-29 EP disclosed
WO-1999050249-A2 PYRIMIDINES AND TRIAZINES AS INTEGRIN ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-10-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010044535-A1 Integrin antagonists ITGB3, VCAM1, ITGB2 KMO 3623/4885EGFR 449/4885ERBB2 161/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.