SCHEMBL7428248

SCHEMBL7428248

Nc1ccc(C[C@H](NC(=O)c2c(Cl)cncc2Cl)C(=O)O)cc1

nearest known ligand 0.76

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 17/20 0.76
ITGB1 P05556 17/20 0.76
ITGB7 P26010 4/20 0.56
ITGA5 P08648 2/20 0.54
ITGB3 P05106 1/20 0.54
ITGAV P06756 1/20 0.54
CA2 P00918 1/20 0.53
ITGA2 P17301 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736989 0.88 ITGA4 (0.77) ITGA4ITGB1ITGB7ITGA5ITGB3
SCHEMBL181376 0.87 ITGB1 (0.65) ITGA4ITGB1ITGB7ITGA5ITGAV
SCHEMBL181378 0.87 ITGB1 (0.65) ITGA4ITGB1ITGB7ITGA5ITGAV
SCHEMBL7428016 0.86 ITGA4 (0.58) ITGA4ITGB1ITGB7ITGA5ITGB3
Hydrochloric Acid SCHEMBL6510331 0.85 ITGA4 (0.57) ITGA4ITGB1ITGB7ITGA5ITGB3
SCHEMBL21376626 0.83 ITGA4 (0.55) ITGA4ITGB1ITGB7ITGA5ITGB3
SCHEMBL7906199 0.81 ITGA4 (0.53) ITGA4ITGB1ITGB7ITGA5ITGB3
SCHEMBL7538961 0.79 ITGB1 (0.73) ITGA4ITGB1ITGB7ITGA5ITGAV
SCHEMBL28742822 0.78 ITGB1 (0.56) ITGA4ITGB1ITGB7ITGA5ITGA2
SCHEMBL28742820 0.78 ITGB1 (0.56) ITGA4ITGB1ITGB7ITGA5ITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082294-A1 PHENYLALANINE DERIVATIVES AS INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2001-03-14 EP claimed
WO-1999064390-A1 PHENYLALANINE DERIVATIVES AS INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 1999-12-16 WO claimed
US-20020035127-A1 Phenylalanine derivatives CELLTECH THERAPEUTIS, LIMITED 2002-03-21 US disclosed
US-6329372-B1 HETEROCYCLIC AMIDE COMPOUNDS ARE ABLE TO INHIBIT THE BINDING OF ALPHA4 INTEGRINS TO THEIR LIGANDS AND ARE OF USE IN THE PROPHYLAXIS AND TREATMENT OF IMMUNE OR INFLAMMATORY DISORDERS. CELLTECH THERAPEUTICS LIMITED (GB) 2001-12-11 US disclosed
EP-1082294-A1 PHENYLALANINE DERIVATIVES AS INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2001-03-14 EP disclosed
WO-1999064390-A1 PHENYLALANINE DERIVATIVES AS INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 1999-12-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020035127-A1 Phenylalanine derivatives PAH, VCAM1, IL4I1 ITGA4 5/4885ITGB1 8/4885ITGB7 25/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.