SCHEMBL7428261

SCHEMBL7428261

COc1ccc([CH]OC2CCCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
KMT2A Q03164 1/20 0.44
NFE2L2 Q16236 1/20 0.44
ALDH1A1 P00352 3/20 0.44
CYP2A6 P11509 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
CHRNA7 P36544 1/20 0.41
TRPA1 O75762 1/20 0.41
RELA Q04206 1/20 0.41
CYP1A2 P05177 1/20 0.41
CA12 O43570 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21596594 0.81 TRPM8 (0.50) RAB9ANPC1NFE2L2ALDH1A1TRPM8
SCHEMBL23244052 0.81 TRPM8 (0.50) RAB9ANPC1NFE2L2ALDH1A1TRPM8
SCHEMBL8321392 0.77 RAB9A (0.42) RAB9ANPC1KMT2ANFE2L2ALDH1A1
SCHEMBL1004985 0.76 POLB (0.41) KDM4EMAPTHPGDCYP3A4CHRNA7
SCHEMBL1006660 0.75 IDO1 (0.43) TRPM8KDM4EMAPTHPGDCYP3A4
SCHEMBL1071370 0.74 MAPT (0.53) RAB9AKMT2AALDH1A1KDM4EMAPT
SCHEMBL3148517 0.72 MAPT (0.51) RAB9ANPC1KMT2AALDH1A1KDM4E
SCHEMBL1156837 0.71 ALDH1A1 (0.58) RAB9ANPC1NFE2L2ALDH1A1CYP2A6
SCHEMBL600597 0.69 HTT (0.70) RAB9AKMT2ATRPM8MAPTLMNA
SCHEMBL154420 0.69 HTT (0.70) RAB9AKMT2ATRPM8MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799040-A4 TRISUBSTITUTED THIOXANTHINES EURO CELTIQUE SA (LU) 1998-04-01 EP claimed
EP-0799040-A1 TRISUBSTITUTED THIOXANTHINES Euroceltique S.A. (LU) 1997-10-08 EP claimed
WO-1996018400-A1 TRISUBSTITUTED THIOXANTHINES EURO-CELTIQUE, S.A. (LU) 1996-06-20 WO claimed