SCHEMBL7443752

SCHEMBL7443752

COc1cc2c(C)nc(OC(=O)N3CCNCC3)c([N+](=O)[O-])c2cc1OC

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
MAPT P10636 3/20 0.36
BLM P54132 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 2/20 0.35
APAF1 O14727 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
UBE2N P61088 1/20 0.35
PDGFRB P09619 2/20 0.35
KIT P10721 1/20 0.35
PDGFRA P16234 1/20 0.35
FLT3 P36888 1/20 0.35
PKM P14618 2/20 0.34
CCNT1 O60563 1/20 0.34
CDK9 P50750 1/20 0.34
CFTR P13569 2/20 0.33
NCF1 P14598 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432960 0.86 KCNH2 (0.44) KDM4EMAPTALDH1A1CCNT1CDK9
SCHEMBL7439631 0.80 MAPT (0.40) KDM4EMAPTBLMTDP1ALDH1A1
SCHEMBL7437559 0.76 KMT2A (0.41) KDM4EMAPTBLMTDP1ALDH1A1
SCHEMBL7441183 0.74 LMNA (0.39) KDM4EMAPTBLMTDP1ALDH1A1
SCHEMBL7446369 0.73 MEN1 (0.40) KDM4EMAPTTDP1ALDH1A1POLB
SCHEMBL7428283 0.72 VCP (0.39) KDM4EMAPTBLMTDP1ALDH1A1
SCHEMBL7440312 0.71 NCEH1 (0.40) KDM4EALDH1A1
SCHEMBL7444737 0.71 PDE3B (0.44) MAPTALDH1A1APAF1
SCHEMBL25301661 0.70 EPHX2 (0.48) KDM4EMAPTTDP1ALDH1A1HPGD
SCHEMBL7412702 0.70 KDM4E (0.44) KDM4EMAPTBLMTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4880817-A O-functionalized derivatives of substituted isoquinolin-3-ols having cardiotonic and/or phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-11-14 US disclosed