SCHEMBL7428568

SCHEMBL7428568

CC(C)(C)C(=O)OCc1cc2cccc(C(=O)O)c2[nH]1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 1/20 0.52
GLA P06280 1/20 0.52
DHODH Q02127 1/20 0.45
KDM5A P29375 5/20 0.41
KDM5B Q9UGL1 4/20 0.41
KDM4A O75164 1/20 0.40
KEAP1 Q14145 1/20 0.39
KDM4C Q9H3R0 10/20 0.39
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
NPC1 O15118 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421572 0.86 ALDH1A1 (0.47) KDM4EALDH1A1GLA
SCHEMBL13492005 0.78 DHODH (0.54) KDM4EDHODHKDM5AKDM5BKDM4A
SCHEMBL4433221 0.77 MTNR1A (0.49) KDM4EALDH1A1GLAMTNR1AMTNR1B
SCHEMBL27285942 0.73 KDM5A (0.49) DHODHKDM5AKDM5BKEAP1MTNR1A
SCHEMBL7648523 0.72 KDM5B (0.60) KDM4EDHODHKDM5AKDM5BKDM4A
SCHEMBL13491530 0.72 DHODH (0.54) KDM4EALDH1A1DHODHKDM5AKDM5B
SCHEMBL10990305 0.71 KDM5A (0.47) DHODHKDM5AKDM5B
SCHEMBL10981682 0.71 KDM5A (0.47) DHODHKDM5AKDM5B
SCHEMBL10982575 0.71 KDM5A (0.47) DHODHKDM5AKDM5B
SCHEMBL2078975 0.70 DHODH (0.58) KDM4EALDH1A1DHODHKEAP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946519-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-06 EP disclosed
WO-1998024771-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-06-11 WO disclosed