SCHEMBL7429456

SCHEMBL7429456

O=C(O)C(Cc1ccccc1)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
TP53 P04637 1/20 0.53
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MMP2 P08253 1/20 0.52
P4HTM Q9NXG6 1/20 0.51
CPA1 P15085 3/20 0.50
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
EPHX1 P07099 1/20 0.50
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
ANPEP P15144 1/20 0.47
ERAP2 Q6P179 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6810144 0.94 KMT2A (0.52) NPC1RAB9ASMN1; SMN2TP53MEN1
SCHEMBL6810226 0.94 KMT2A (0.52) NPC1RAB9ASMN1; SMN2TP53MEN1
SCHEMBL27581400 0.88 NPC1 (0.54) NPC1RAB9ASMN1; SMN2TP53MEN1
SCHEMBL6625969 0.88 EPHX1 (0.69) NPC1RAB9ASMN1; SMN2TP53MEN1
SCHEMBL2658881 0.83 ALDH1A1 (0.48) NPC1RAB9ASMN1; SMN2TP53MEN1
Toluene SCHEMBL28163126 0.83 RAB9A (0.45) NPC1RAB9ASMN1; SMN2TP53MEN1
SCHEMBL27581401 0.82 ESR1 (0.54) NPC1RAB9ASMN1; SMN2TP53MEN1
Nitrobenzene SCHEMBL28691684 0.81 AKR1C3 (0.58) NPC1MEN1KMT2ACRHBPCRHR2
SCHEMBL599399 0.81 EPHX1 (0.71) P4HTMCPA1EPHX1CYP1A2CYP2C19
SCHEMBL67234 0.81 EPHX1 (0.71) P4HTMCPA1EPHX1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105330630-B Benzofuran compounds and its preparation method and application 上海交通大学 2018-04-17 CN disclosed
US-9718763-B2 Catalytic ester decarbonylation REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2017-08-01 US disclosed
US-20160194276-A1 CATALYTIC ESTER DECARBONYLATION REGENTS OF THE UNIVERSITY OF MINNESOTA 2016-07-07 US disclosed
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed
US-4520007-A Anti-coagulants of the 4-hydroxycoumarin type and rodenticidal compositions (baits) comprising such anti-coagulants SHELL OIL COMPANY (US) 1985-05-28 US disclosed
EP-0098629-A1 Anti-coagulants of the 4-hydroxycoumarin type, the preparation thereof, and rodenticidal compositions (baits) comprising such anti-coagulants SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1984-01-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160194276-A1 CATALYTIC ESTER DECARBONYLATION DECR1, C1S, CBR3 NPC1 2770/4885RAB9A 2853/4885SMN1; SMN2 3519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.