SCHEMBL7429615

SCHEMBL7429615

CCN1C(C)=C(C(=O)O)C(CC)(c2cccc([N+](=O)[O-])c2)C(C(=O)O)=C1C#N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 4/20 0.37
LMNA P02545 3/20 0.37
KDM4E B2RXH2 3/20 0.37
KMT2A Q03164 2/20 0.37
TP53 P04637 1/20 0.36
MAPT P10636 4/20 0.34
NPSR1 Q6W5P4 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TSHR P16473 2/20 0.34
PTBP1 P26599 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
NFKB1 P19838 1/20 0.34
CYP2C19 P33261 1/20 0.34
GMNN O75496 1/20 0.34
BLM P54132 1/20 0.34
PMP22 Q01453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10874214 0.84 TDP1 (0.38) TDP1ALDH1A1LMNAKDM4EKMT2A
SCHEMBL10872894 0.83 TDP1 (0.38) TDP1ALDH1A1LMNAKMT2ATP53
SCHEMBL4883866 0.82 TP53 (0.43) TDP1ALDH1A1LMNAKMT2ATP53
SCHEMBL4756165 0.79 TP53 (0.43) TDP1ALDH1A1LMNAKMT2ATP53
SCHEMBL10567035 0.78 SIGMAR1 (0.43) TDP1ALDH1A1LMNAKDM4EKMT2A
SCHEMBL8295139 0.77 ALDH1A1 (0.39) TDP1ALDH1A1LMNAKDM4EKMT2A
SCHEMBL3392997 0.76 TDP1 (0.40) TDP1ALDH1A1LMNAKDM4EKMT2A
SCHEMBL7439133 0.75 TDP1 (0.38) TDP1ALDH1A1LMNAKMT2ATP53
SCHEMBL8827906 0.75 ALDH1A1 (0.39) ALDH1A1LMNAKDM4EKMT2ATP53
SCHEMBL4758254 0.74 HCAR3 (0.39) TDP1ALDH1A1LMNAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP disclosed
US-4145432-A 6-ACYLORYALKYL-1,4-DIHYDROPYRIDINE DERIVATIVES AND A METHOD OF EFFECTING VASODILATION THEREWITH FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1979-03-20 US disclosed