SCHEMBL7430899

SCHEMBL7430899

COC(=O)[C@H](Cc1ccc(OC)cc1)NC(=O)N(C)CC(O)CO

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
THRB P10828 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD17B10 Q99714 1/20 0.44
REN P00797 1/20 0.42
MMP1 P03956 3/20 0.42
MMP7 P09237 2/20 0.42
MMP8 P22894 2/20 0.42
MMP12 P39900 2/20 0.42
MMP13 P45452 2/20 0.42
LDHA P00338 1/20 0.42
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
MMP3 P08254 1/20 0.40
MMP9 P14780 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431334 0.91 KMT2A (0.50) ALDH1A1RENLDHAKMT2AFPR2
SCHEMBL9832460 0.82 LDHA (0.50) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL9833395 0.82 GAA (0.46) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL16879017 0.78 LDHA (0.54) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL16879018 0.78 LDHA (0.54) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL7292751 0.78 KMT2A (0.55) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL7436585 0.78 MMP1 (0.45) CYP2C19MMP1MMP7MMP8MMP12
SCHEMBL7296180 0.77 REN (0.43) ALDH1A1RENLDHAGAARAB9A
SCHEMBL9833056 0.76 REN (0.45) RENMMP1MMP7MMP8MMP13
SCHEMBL5706152 0.76 ACACB (0.58) ALDH1A1THRBCYP2C9CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0416393-A1 Peptidyl difluorodiol renin inhibitors ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
EP-0258289-A4 PEPTIDE ANALOGS 1991-01-02 EP disclosed
US-4977277-A INTERMEDIATES FOR RENIN INHIBITORS ABBOTT LABORATORIES (US) 1990-12-11 US disclosed
US-4857507-A HYPOTENSIVE AGENT ABBOTT LABORATORIES (US) 1989-08-15 US disclosed
EP-0258289-A1 PEPTIDE ANALOGS ABBOTT LABORATORIES (US) 1988-03-09 EP disclosed
WO-1987004349-A1 PEPTIDE ANALOGS DELLARIA JOSEPH 1987-07-30 WO disclosed