SCHEMBL7432503

SCHEMBL7432503

CCN(CC)C(=O)C1CCCN(CCC(=O)c2ccc(O)c(O)c2[N+](=O)[O-])C1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.49
MAPT P10636 2/20 0.49
MAPK1 P28482 1/20 0.49
LMNA P02545 1/20 0.48
KDM4E B2RXH2 6/20 0.48
BCHE P06276 1/20 0.47
GAA P10253 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.44
HSD17B10 Q99714 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423482 0.83 ALDH1A1 (0.51) ALDH1A1MAPTLMNAKDM4EGAA
SCHEMBL7432684 0.80 ALDH1A1 (0.43) ALDH1A1HSD17B10
SCHEMBL7428303 0.78 ALDH1A1 (0.46) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL7427756 0.77 KMT2A (0.46) ALDH1A1MAPTKDM4EGAAHTT
SCHEMBL7432258 0.77 HTR1A (0.42) ALDH1A1MAPTLMNAKDM4EGAA
SCHEMBL7433195 0.75 KMT2A (0.43) ALDH1A1KDM4ERAB9APOLB
SCHEMBL7434299 0.72 KMT2A (0.48) ALDH1A1MAPTLMNAHTT
SCHEMBL7433801 0.72 DRD2 (0.42)
Bromide SCHEMBL10779800 0.71 BCHE (0.76) ALDH1A1MAPTKDM4EBCHEHTT
SCHEMBL7517410 0.70 ALPL (0.46) ALDH1A1MAPTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020037931-A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them PORTELA & C.A., S.A. (PT) 2002-03-28 US claimed
EP-1167341-A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them Portela & Ca., S.A. (PT) 2002-01-02 EP claimed
WO-2001098250-A1 SUBSTITUTED NITRATED CATECHOLS, THEIR USE IN THE TREATMENT OF SOME CENTRAL AND PERIPHERAL NERVOUS SYSTEM DISORDERS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PORTELA & CA SA (PT) 2001-12-27 WO claimed
US-20020037931-A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them PORTELA & C.A., S.A. (PT) 2002-03-28 US disclosed
EP-1167341-A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them Portela & Ca., S.A. (PT) 2002-01-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020037931-A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them SLC6A2, COMT, SLC6A3 ALDH1A1 477/4885MAPT 379/4885MAPK1 1779/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.