SCHEMBL7434156

SCHEMBL7434156

CC(=O)NC(Cc1ccc(Br)cc1)C(O)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.52
CYP1A2 P05177 1/20 0.47
MME P08473 4/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
FPR2 P25090 2/20 0.42
CTRB1 P17538 4/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7436643 0.86 SLC7A5 (0.51) MMECTRB1
SCHEMBL7441034 0.86 ACACB (0.51) ACACBPPARGPPARACTRB1MEN1
SCHEMBL7434134 0.86 CTRB1 (0.55) CYP1A2CTRB1CTSSCTSKNPC1
SCHEMBL7442013 0.86 CTRB1 (0.55) CYP1A2CTRB1CTSSCTSKNPC1
SCHEMBL7444226 0.85 ALDH1A1 (0.44) PPARGPPARACTRB1CTSSCTSK
SCHEMBL7436512 0.84 ACACB (0.53) ACACBPPARGPPARACTRB1
SCHEMBL7438864 0.84 ACACB (0.56) ACACBMMECTRB1
SCHEMBL7432787 0.82 LDHA (0.58) ACACBPPARGPPARAFPR2KMT2A
SCHEMBL7439954 0.82 LDHA (0.58) ACACBPPARGPPARAFPR2KMT2A
SCHEMBL7438493 0.81 ALDH1A1 (0.46) ACACBPPARANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed