SCHEMBL7434291

SCHEMBL7434291

Nc1cc(Br)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
KDM4E B2RXH2 4/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
MAPT P10636 2/20 0.57
HPGD P15428 3/20 0.50
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
NFKB1 P19838 1/20 0.50
HTT P42858 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
GAA P10253 1/20 0.47
AHR P35869 3/20 0.45
ADORA3 P0DMS8 4/20 0.44
ADORA2A P29274 3/20 0.43
LMNA P02545 1/20 0.43
ADORA1 P30542 2/20 0.42
CYP11B2 P19099 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7428728 0.86 ALDH1A1 (0.43) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7431271 0.84 AMY1A (0.50) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7423524 0.84 ALDH1A1 (0.53) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7438035 0.80 ADORA2A (0.59) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7487566 0.80 KDM4E (0.40) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7428936 0.80 SMN1; SMN2 (0.44) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7483266 0.80 ALDH1A1 (0.43) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL6870681 0.79 ADORA2A (0.49) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7709122 0.78 MAOA (0.47) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL7427474 0.78 SMN1; SMN2 (0.47) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed