SCHEMBL7428728

SCHEMBL7428728

Nc1cc(Br)cc2nc(-c3ccncc3)nn12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 2/20 0.42
HPGD P15428 2/20 0.42
AHR P35869 3/20 0.41
CYP11B2 P19099 1/20 0.41
TP53 P04637 1/20 0.37
CYP2C19 P33261 1/20 0.37
CDC7 O00311 1/20 0.36
MAPK13 O15264 1/20 0.36
DAPK3 O43293 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
PIM1 P11309 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7434291 0.86 ALDH1A1 (0.57) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL7427474 0.79 SMN1; SMN2 (0.47) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL7487566 0.78 KDM4E (0.40) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL7429024 0.76 ADORA2A (0.39) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL7543025 0.75 ADORA2A (0.41) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL7480280 0.75 ADORA2A (0.59) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL7438035 0.75 ADORA2A (0.59) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL7490670 0.74 ADORA2A (0.62) ADORA2A
SCHEMBL7428889 0.72 ADORA2A (0.44) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL7427470 0.72 ADORA2A (0.59) ADORA2ACSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed