SCHEMBL7434679

SCHEMBL7434679

O[C@@H](c1ccccc1)C(Cl)(Cl)Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.47
TSHR P16473 3/20 0.43
LMNA P02545 5/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
MAPK1 P28482 1/20 0.42
SLC6A4 P31645 1/20 0.42
ADRA2C P18825 2/20 0.41
CHRM2 P08172 1/20 0.41
ADRA1A P35348 1/20 0.41
RGS12 O14924 1/20 0.41
GLA P06280 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
NFKB1 P19838 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4372186 1.00 AOC3 (0.47) AOC3TSHRLMNACES2CES1
SCHEMBL23172374 1.00 AOC3 (0.47) AOC3TSHRLMNACES2CES1
Acetic Acid SCHEMBL7640545 0.89 HPGD (0.46) AOC3LMNACES2CES1MAPK1
Alcohol SCHEMBL10526338 0.89 LMNA (0.48) AOC3TSHRLMNASLC6A4ADRA2C
SCHEMBL30387499 0.82 AOC3 (0.45) AOC3TSHRLMNACES2CES1
SCHEMBL11150798 0.82 AOC3 (0.45) AOC3TSHRLMNACES2CES1
SCHEMBL23149900 0.81 SRD5A2 (0.50) TSHR
SCHEMBL10525043 0.80 CYP2D6 (0.41) AOC3LMNASLC6A4ADRA1ACYP3A4
SCHEMBL76211 0.77 TSHR (0.58) AOC3TSHRLMNAMAPK1CYP2D6
SCHEMBL7120983 0.77 ESR1 (0.62) TSHRLMNACHRM2ADRA1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11570987-B2 Pesticidal compounds and methods of use NEW YORK UNIVERSITY (US) 2023-02-07 US disclosed
US-20210092950-A1 PESTICIDAL COMPOUNDS AND METHODS OF USE NEW YORK UNIVERSITY (US) 2021-04-01 US disclosed
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
EP-0458823-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES. BOEHRINGER MANNHEIM ITALIA (IT) 1991-12-04 EP disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed
US-4686217-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS FISONS PLC (GB) 1987-08-11 US disclosed
US-4607041-A CARDIOTONIC AGENTS FISONS PLC (GB) 1986-08-19 US disclosed
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210092950-A1 PESTICIDAL COMPOUNDS AND METHODS OF USE ACHE, DDT, PTMS AOC3 1566/4885TSHR 2895/4885LMNA 2786/4885
US-11570987-B2 Pesticidal compounds and methods of use ACHE, DDT, PTMS AOC3 1566/4885TSHR 2895/4885LMNA 2786/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.