SCHEMBL7120983

SCHEMBL7120983

Oc1ccc(C(O)C(Cl)(Cl)Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.62
ESR2 Q92731 7/20 0.62
PDCD1 Q15116 1/20 0.44
CD274 Q9NZQ7 1/20 0.44
TAAR1 Q96RJ0 3/20 0.43
HIF1A Q16665 3/20 0.43
NFKB1 P19838 2/20 0.43
HTR3A P46098 1/20 0.43
TSHR P16473 1/20 0.43
ALOX15 P16050 3/20 0.41
KDM4E B2RXH2 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
APEX1 P27695 1/20 0.41
CYP3A4 P08684 3/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
THPO P40225 2/20 0.40
BLM P54132 2/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL76211 0.80 TSHR (0.58) ESR1ESR2HIF1ATSHRALOX15
SCHEMBL23149894 0.78 AOC3 (0.38) ESR1ESR2HIF1ATSHRKDM4E
SCHEMBL23149874 0.78 AOC3 (0.38) ESR1ESR2HIF1ATSHRKDM4E
SCHEMBL23149895 0.78 AOC3 (0.38) ESR1ESR2HIF1ATSHRKDM4E
SCHEMBL11302427 0.78 HPGD (0.44) ESR1ESR2HIF1ATSHRTDP1
SCHEMBL23172374 0.77 AOC3 (0.47) NFKB1TSHRALOX15KDM4ECYP3A4
SCHEMBL7434679 0.77 AOC3 (0.47) NFKB1TSHRALOX15KDM4ECYP3A4
SCHEMBL4372186 0.77 AOC3 (0.47) NFKB1TSHRALOX15KDM4ECYP3A4
SCHEMBL8580685 0.77 ESR1 (0.65) ESR1ESR2PDCD1CD274TAAR1
SCHEMBL44658 0.77 ESR1 (1.00) ESR1ESR2PDCD1CD274TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030144541-A1 Process for preparing alpha-halogenated retones RHODIA CHIMIE (FR) 2003-07-31 US claimed
EP-1250303-A1 METHOD FOR PREPARING ALPHA-HALOGENATED KETONES RHODIA CHIMIE (FR) 2002-10-23 EP claimed
WO-2001055067-A1 METHOD FOR PREPARING ALPHA-HALOGENATED KETONES RHODIA CHIMIE (FR) 2001-08-02 WO claimed
US-4249015-A Preparation of organic acids and/or esters SHELL OIL COMPANY (US) 1981-02-03 US claimed
JP-58052236-A None JP disclosed
JP-56016464-A None JP disclosed
US-20030144541-A1 Process for preparing alpha-halogenated retones RHODIA CHIMIE (FR) 2003-07-31 US disclosed
EP-1250303-A1 METHOD FOR PREPARING ALPHA-HALOGENATED KETONES RHODIA CHIMIE (FR) 2002-10-23 EP disclosed
WO-2001055067-A1 METHOD FOR PREPARING ALPHA-HALOGENATED KETONES RHODIA CHIMIE (FR) 2001-08-02 WO disclosed
US-4544766-A HYDROLYSIS OF DICHLOROETHENYL COMPOUND OTSUKA KAGAKU YAKUHIN KABUSHIKI KAISHA (JP) 1985-10-01 US disclosed
US-4504678-A Pure crystalline racemic sodium parahydroxymandelate, process for its preparation and uses thereof SOCIETE FRANCAISE HOECHST (FR) 1985-03-12 US disclosed
US-4408070-A SODIUM P-FORMYLPHENOLATE SOCOETE FRANCAISE HOECHST (FR) 1983-10-04 US disclosed
JP-S5852236-A DICHLOROSTYRENE DERIVATIVE AND ITS PREPARATION SHIYOUNO TAMIE 1983-03-28 JP disclosed
JP-S5616464-A PRODUCTION OF ALPHA-METHYLTHIO-4-HYDROXYPHENYLACETIC ACID NIPPON SODA CO LTD 1981-02-17 JP disclosed
US-4249015-A Preparation of organic acids and/or esters SHELL OIL COMPANY (US) 1981-02-03 US disclosed
US-4105857-A CONDENSING PHENOL AND CHLORAL IN A SULFURIC ACID- METHYLENE CHLORIDE SOLVENT SYSTEM GENERAL ELECTRIC COMPANY (US) 1978-08-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030144541-A1 Process for preparing alpha-halogenated retones ADH1A, ADH1C, RER1 ESR1 1300/4885ESR2 765/4885PDCD1 3152/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.