SCHEMBL7434800

SCHEMBL7434800

Cc1cccc(-c2c[nH]c(C(N)=NOS(C)(=O)=O)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 2/20 0.41
ATP4A P20648 2/20 0.39
ATP4B P51164 2/20 0.39
XDH P47989 1/20 0.39
SDHB P21912 1/20 0.38
KMO O15229 2/20 0.36
PIN1 Q13526 1/20 0.36
IDO1 P14902 1/20 0.35
METAP2 P50579 1/20 0.35
ICMT O60725 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
DHODH Q02127 1/20 0.34
PKM P14618 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA5A P35218 1/20 0.34
CA5B Q9Y2D0 1/20 0.34
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426997 0.88 MAPT (0.36) SLC9A1ALDH1A1MAPT
SCHEMBL7440169 0.87 SLC9A1 (0.41) SLC9A1KMOIDO1ICMTPKM
SCHEMBL7440591 0.85 ALPL (0.35) SLC9A1NPC1RAB9APKMPTGS1
SCHEMBL7438866 0.77 SCN9A (0.41) SLC9A1ATP4AATP4BXDHSDHB
SCHEMBL7433733 0.77 DHODH (0.48) SLC9A1ATP4AATP4BXDHKMO
SCHEMBL7434796 0.72 SLC9A1 (0.41) SLC9A1ATP4AATP4BXDHSDHB
SCHEMBL7489817 0.70 JAK2 (0.52) KMONPC1RAB9AALDH1A1MAPT
SCHEMBL10604269 0.66 IDO1 (0.51) ATP4AATP4BXDHKMOIDO1
SCHEMBL7433050 0.65 SCN9A (0.43) SLC9A1KMOPTGS1PTGS2MAPT
SCHEMBL29662867 0.65 MAPK14 (0.56) SDHBCA1CA2PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0506194-B1 4-aryl-thiazole or imidazole derivatives AKZO NOBEL NV (NL) 1996-08-21 EP disclosed
US-5462959-A 4-aryl-imidazole derivatives AKZO N.V. (NL) 1995-10-31 US disclosed
US-5254575-A 4-aryl-thiazole derivatives AKZO N.V. (NL) 1993-10-19 US disclosed
EP-0506194-A1 4-aryl-thiazole or imidazole derivatives Akzo Nobel N.V. (NL) 1992-09-30 EP disclosed