SCHEMBL7435251

SCHEMBL7435251

O=[C]c1cc(-c2ccccc2)c(=O)n2c1-c1cc(Cl)ccc1CC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.38
F7 P08709 1/20 0.35
PARP1 P09874 1/20 0.35
F3 P13726 1/20 0.35
PARP10 Q53GL7 1/20 0.35
NPY5R Q15761 1/20 0.34
KMT2A Q03164 4/20 0.33
GABRA1 P14867 3/20 0.33
GABRG2 P18507 3/20 0.33
GABRB3 P28472 3/20 0.33
GABRA3 P34903 3/20 0.33
GABRA2 P47869 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
OPRK1 P41145 3/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
CACNA1F O60840 1/20 0.33
ALB P02768 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9335056 0.83 GABRA1 (0.36) CNR1F7PARP1F3PARP10
SCHEMBL9335063 0.83 GABRA1 (0.40) F7PARP1F3PARP10NPY5R
SCHEMBL8936714 0.81 HSP90AA1 (0.38) KMT2AKDM4EMAPTNPSR1ALDH1A1
SCHEMBL9338054 0.81 HSD17B3 (0.38) CNR1F7PARP1F3PARP10
SCHEMBL27273993 0.81 PDE10A (0.43) PARP1KDM4EMAPTNPSR1OPRK1
SCHEMBL7284938 0.79 MAPT (0.40) F7PARP1F3PARP10NPY5R
SCHEMBL9338217 0.78 ACHE (0.35) CNR1NPY5RKMT2AGABRA1GABRG2
SCHEMBL10369849 0.77 HSD17B3 (0.37) KMT2AGABRA1GABRG2GABRB3GABRA3
SCHEMBL9334812 0.77 GABRA1 (0.48) CNR1KMT2AGABRA1GABRG2GABRB3
SCHEMBL9334794 0.77 TSHR (0.41) KDM4EALDH1A1SMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0650966-A1 Process for the preparation of a benzo(a)quinolizinone derivative F. HOFFMANN-LA ROCHE AG (CH) 1995-05-03 EP disclosed