SCHEMBL27273993

SCHEMBL27273993

COc1cc(-c2ccccc2)c(=O)n2c1-c1cc(Cl)ccc1CC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 5/20 0.43
PDE7A Q13946 2/20 0.43
PDE3A Q14432 2/20 0.43
ACHE P22303 1/20 0.42
KDM4E B2RXH2 4/20 0.39
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
ALDH1A1 P00352 5/20 0.37
GPR84 Q9NQS5 3/20 0.37
GAA P10253 2/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B3 P37058 1/20 0.37
GLA P06280 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PARP1 P09874 1/20 0.37
PRMT5 O14744 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10367806 0.87 ALDH1A1 (0.38) PDE10APDE7APDE3AACHEKDM4E
SCHEMBL7284938 0.87 MAPT (0.40) PDE10APDE7APDE3AACHEKDM4E
SCHEMBL9335063 0.85 GABRA1 (0.40) KDM4EOPRK1MAPTHSD17B3PARP1
SCHEMBL9338217 0.84 ACHE (0.35) PDE10APDE7APDE3AACHEKDM4E
SCHEMBL9334812 0.83 GABRA1 (0.48) KDM4EALDH1A1GAAMAPTHSD17B3
SCHEMBL9335056 0.82 GABRA1 (0.36) PDE3AKDM4EOPRK1ALDH1A1GAA
SCHEMBL7435251 0.81 CNR1 (0.38) KDM4EOPRK1ALDH1A1GAAMAPT
SCHEMBL9338054 0.81 HSD17B3 (0.38) KDM4EMAPTHSD17B3MAPK1PARP1
SCHEMBL8936714 0.81 HSP90AA1 (0.38) KDM4EALDH1A1GAAMAPTHSD17B3
SCHEMBL9338273 0.80 ACHE (0.36) ACHEKDM4EOPRK1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1016871-B Process for the preparation of bicyclic and tricyclic pyridine derivatives HOFFMANN LA ROCHE 7 CO F (CN) 1992-06-03 CN disclosed