SCHEMBL7435308

SCHEMBL7435308

CSCC(=O)C(CCc1ccccc1)NCCCC(C)N(C)C(=O)COc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ALOX5 P09917 1/20 0.40
HDAC8 Q9BY41 1/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
POLB P06746 1/20 0.37
SIGMAR1 Q99720 1/20 0.36
MAPK1 P28482 1/20 0.36
GGT1 P19440 1/20 0.35
PTPN1 P18031 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301637 0.85 ALDH1A1 (0.44) SMN1; SMN2NPC1RAB9AALOX5ALDH1A1
SCHEMBL7303790 0.78 ALDH1A1 (0.44) SMN1; SMN2NPC1RAB9AHDAC8ALDH1A1
SCHEMBL7311207 0.77 ALDH1A1 (0.45) SMN1; SMN2NPC1RAB9AALDH1A1MEN1
SCHEMBL7302476 0.76 MAPT (0.44) SMN1; SMN2NPC1RAB9AALDH1A1KMT2A
SCHEMBL7435291 0.73 CTSL (0.50) ALDH1A1POLB
SCHEMBL7435315 0.73 CTSL (0.50) ALDH1A1POLB
SCHEMBL7309575 0.71 ALDH1A1 (0.41) SMN1; SMN2ALDH1A1MEN1KMT2APOLB
SCHEMBL7307305 0.70 MAPT (0.36) SMN1; SMN2ALDH1A1POLB
SCHEMBL7313893 0.70 MAPT (0.36) SMN1; SMN2ALDH1A1MEN1KMT2APOLB
SCHEMBL7302949 0.70 POLB (0.43) HDAC8MEN1KMT2APOLBPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed