SCHEMBL7435408

SCHEMBL7435408

COc1ccc(C(=O)C(NC(C)=O)C(O)C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
CYP1A2 P05177 1/20 0.51
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
ACACB O00763 1/20 0.43
PLK1 P53350 1/20 0.42
MAPT P10636 2/20 0.42
POLB P06746 1/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
SLC2A1 P11166 1/20 0.42
HPGD P15428 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
PARP1 P09874 1/20 0.41
PARP10 Q53GL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437066 0.86 KMT2A (0.51) ALDH1A1ACACBMAPTPOLBNPC1
SCHEMBL7485958 0.85 NPSR1 (0.54) CYP1A2ACACBPLK1MAPTMEN1
SCHEMBL7442141 0.83 NPC1 (0.49) ALDH1A1CES2CES1MEN1NPC1
SCHEMBL7496442 0.83 LMNA (0.40) ALDH1A1CA1CA2CES2MAPT
SCHEMBL7434063 0.83 CES2 (0.43) ALDH1A1CES2CES1MAPTKMT2A
SCHEMBL7500101 0.82 NPC1 (0.41) ALDH1A1CA1CA2CES2CES1
SCHEMBL7430292 0.82 CYP1A2 (0.49) ALDH1A1CYP1A2CES2CES1ACACB
SCHEMBL7495222 0.81 ACACB (0.48) ACACBMAPTMEN1KMT2A
SCHEMBL7436814 0.81 SMN1; SMN2 (0.47) ALDH1A1ACACBMAPTNPC1RAB9A
SCHEMBL7497110 0.79 ALDH1A1 (0.46) ALDH1A1ACACBPLK1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed