SCHEMBL7430292

SCHEMBL7430292

CC(=O)NC(C(=O)c1ccc(Br)cc1)C(O)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
LMNA P02545 3/20 0.42
ALDH1A1 P00352 3/20 0.41
FPR2 P25090 4/20 0.40
CA12 O43570 1/20 0.38
MMP2 P08253 1/20 0.38
CA14 Q9ULX7 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
GAA P10253 1/20 0.38
UBE2N P61088 1/20 0.38
ACACB O00763 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
KMT2A Q03164 3/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 2/20 0.37
NPC1 O15118 1/20 0.37
CYP3A4 P08684 1/20 0.37
NFKB1 P19838 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7496442 0.86 LMNA (0.40) LMNAALDH1A1CA12CA14CES2
SCHEMBL7434063 0.85 CES2 (0.43) LMNAALDH1A1SMN1; SMN2CES2CES1
SCHEMBL7500101 0.84 NPC1 (0.41) ALDH1A1GAACES2CES1KMT2A
SCHEMBL7436814 0.83 SMN1; SMN2 (0.47) LMNAALDH1A1SMN1; SMN2GAAACACB
SCHEMBL7435408 0.82 ALDH1A1 (0.51) CYP1A2ALDH1A1ACACBCES2CES1
SCHEMBL7497110 0.82 ALDH1A1 (0.46) LMNAALDH1A1GAAACACBKMT2A
SCHEMBL7437066 0.80 KMT2A (0.51) LMNAALDH1A1SMN1; SMN2ACACBKMT2A
SCHEMBL7493041 0.80 L3MBTL1 (0.47) LMNAALDH1A1GAAACACBKMT2A
SCHEMBL7490643 0.79 KDM4E (0.50) CYP1A2LMNACA12CA14SMN1; SMN2
SCHEMBL7485958 0.79 NPSR1 (0.54) CYP1A2LMNASMN1; SMN2GAAACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed