SCHEMBL7436334

SCHEMBL7436334

Nc1cc(N2CCOCC2)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
NPSR1 Q6W5P4 4/20 0.47
HSD17B10 Q99714 3/20 0.47
TSHR P16473 3/20 0.47
MAPK1 P28482 3/20 0.47
MAPT P10636 3/20 0.47
GAA P10253 1/20 0.45
HPGD P15428 4/20 0.45
ALDH1A1 P00352 3/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 2/20 0.45
PRKDC P78527 1/20 0.43
LMNA P02545 3/20 0.43
PIK3CA P42336 3/20 0.43
MTOR P42345 2/20 0.43
PIK3R1 P27986 1/20 0.43
MEN1 O00255 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
AR P10275 1/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709059 0.88 SMN1; SMN2 (0.45) HTTHSD17B10TSHRMAPTGAA
SCHEMBL7705992 0.87 HPGD (0.45) HTTHSD17B10TSHRMAPK1MAPT
SCHEMBL7427937 0.83 ADORA2A (0.56) HTTNPSR1MAPK1ALDH1A1KMT2A
SCHEMBL7423524 0.75 ALDH1A1 (0.53) HTTMAPTGAAHPGDALDH1A1
SCHEMBL7434291 0.73 ALDH1A1 (0.57) HTTMAPTGAAHPGDALDH1A1
SCHEMBL7705975 0.72 GBA1 (0.48) GAAKMT2AKDM4EMEN1
SCHEMBL7480538 0.72 ADORA2A (0.65) ALDH1A1ADORA2AADORA1
SCHEMBL7711835 0.71 ADORA2A (0.64) TSHRMAPK1MAPTKMT2AKDM4E
SCHEMBL7430368 0.71 ADORA2A (0.66) ALDH1A1ADORA2AADORA1
SCHEMBL6870681 0.70 ADORA2A (0.49) HTTNPSR1MAPTGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed