SCHEMBL7436514

SCHEMBL7436514

Cn1c(=O)[nH]c(N)c(/N=C/c2ccccc2)c1=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
G6PD P11413 2/20 0.57
LIG1 P18858 2/20 0.55
LIG3 P49916 1/20 0.55
LIG4 P49917 1/20 0.55
CDK1 P06493 1/20 0.48
TPI1 P60174 1/20 0.48
GAA P10253 5/20 0.45
KDM4E B2RXH2 2/20 0.45
GLA P06280 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 4/20 0.41
LMNA P02545 2/20 0.41
PKM P14618 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
MAOB P27338 2/20 0.40
ADORA3 P0DMS8 2/20 0.40
ADORA2B P29275 2/20 0.40
ADORA2A P29274 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4407466 1.00 G6PD (0.57) G6PDLIG1LIG3LIG4CDK1
SCHEMBL7443806 0.80 G6PD (0.53) G6PDLIG1LIG3LIG4GAA
SCHEMBL7443811 0.80 G6PD (0.53) G6PDLIG1LIG3LIG4GAA
SCHEMBL4379825 0.77 ALDH1A1 (0.47) G6PDLIG1LIG3LIG4CDK1
SCHEMBL4379829 0.77 ALDH1A1 (0.47) G6PDLIG1LIG3LIG4CDK1
SCHEMBL1946777 0.74 ALDH1A1 (0.50) CDK1TPI1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL22105776 0.69 G6PD (0.53) G6PDLIG1LIG3LIG4CDK1
SCHEMBL7435188 0.65 GAA (0.52) GAAKDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL21946635 0.64 G6PD (0.68) G6PDLIG1LIG3LIG4CDK1
SCHEMBL1943938 0.64 MEN1 (0.43) G6PDGAAKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939419-A HYPOTENSIVE AGENTS AND BRONCHODILATOR AGENTS SCHERING-PLOUGH CORPORATION (US) 1999-08-17 US disclosed
EP-0538332-B1 POLYCYCLIC GUANINE DERIVATIVES SCHERING CORP (US) 1997-07-23 EP disclosed
EP-0686157-A1 2-BENZYL-POLYCYCLIC GUANINE DERIVATIVES AND PROCESS FOR PREPARING THEM SCHERING CORPORATION (US) 1995-12-13 EP disclosed
US-5393755-A Hypotensive agents, enzyme inhibitors SCHERING CORPORATION (US) 1995-02-28 US disclosed
WO-1994019351-A1 2-BENZYL-POLYCYCLIC GUANINE DERIVATIVES AND PROCESS FOR PREPARING THEM SCHERING CORPORATION (US) 1994-09-01 WO disclosed
WO-1991019717-A1 POLYCYCLIC GUANINE DERIVATIVES SCHERING CORPORATION (US) 1991-12-26 WO disclosed