SCHEMBL7435188

SCHEMBL7435188

CN(c1ccccc1)c1c(N)[nH]c(=O)n(C)c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.52
ADORA2B P29275 3/20 0.41
ADORA3 P0DMS8 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 1/20 0.41
KDM4C Q9H3R0 2/20 0.40
GFER P55789 1/20 0.39
HSD17B10 Q99714 3/20 0.36
KMT2A Q03164 2/20 0.36
NR3C1 P04150 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
MEN1 O00255 1/20 0.36
CASP1 P29466 1/20 0.36
BRCA1 P38398 1/20 0.36
CASP7 P55210 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PKM P14618 1/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 3/20 0.36
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7434385 0.80 ALDH1A1 (0.50) KMT2AMEN1SMN1; SMN2PKMALDH1A1
SCHEMBL7444168 0.69 KMT2A (0.39) GAAKMT2ANR3C1MEN1SMN1; SMN2
SCHEMBL5307352 0.69 GAA (1.00) GAAADORA2BADORA3KDM4CHSD17B10
SCHEMBL9300715 0.68 L3MBTL1 (0.32) GAAADORA2BADORA3ADORA2AADORA1
SCHEMBL4407466 0.65 G6PD (0.57) GAAADORA2BADORA3ADORA2AADORA1
SCHEMBL4406872 0.65 ALDH1A1 (0.53) GAAKMT2ANR3C1MEN1CASP1
SCHEMBL7436514 0.65 G6PD (0.57) GAAADORA2BADORA3ADORA2AADORA1
SCHEMBL1947320 0.65 ADORA2B (0.39) GAAADORA2BADORA3ADORA2AADORA1
SCHEMBL8696414 0.63 TYMP (0.41) GAAADORA2BADORA3ADORA2AADORA1
SCHEMBL21479953 0.62 MEN1 (0.41) GAAKMT2AMEN1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939419-A HYPOTENSIVE AGENTS AND BRONCHODILATOR AGENTS SCHERING-PLOUGH CORPORATION (US) 1999-08-17 US disclosed
EP-0538332-B1 POLYCYCLIC GUANINE DERIVATIVES SCHERING CORP (US) 1997-07-23 EP disclosed
EP-0686157-A1 2-BENZYL-POLYCYCLIC GUANINE DERIVATIVES AND PROCESS FOR PREPARING THEM SCHERING CORPORATION (US) 1995-12-13 EP disclosed
US-5393755-A Hypotensive agents, enzyme inhibitors SCHERING CORPORATION (US) 1995-02-28 US disclosed
WO-1994019351-A1 2-BENZYL-POLYCYCLIC GUANINE DERIVATIVES AND PROCESS FOR PREPARING THEM SCHERING CORPORATION (US) 1994-09-01 WO disclosed
WO-1991019717-A1 POLYCYCLIC GUANINE DERIVATIVES SCHERING CORPORATION (US) 1991-12-26 WO disclosed