SCHEMBL7436797

SCHEMBL7436797

CC(C)(C)OC(=O)CC(N)C(=O)C(C(=O)OCc1ccccc1)n1nnnc1C1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.36
SLC6A4 P31645 1/20 0.36
CTSL P07711 1/20 0.35
ELANE P08246 1/20 0.35
CACNA1B Q00975 4/20 0.35
ALDH1A1 P00352 1/20 0.35
GHSR Q92847 1/20 0.35
FKBP1A P62942 3/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7446446 0.84 CTSL (0.38) HTR2CSLC6A4CTSLALDH1A1GHSR
SCHEMBL7443228 0.84 HTR2C (0.38) HTR2CSLC6A4CTSLCACNA1BFKBP1A
SCHEMBL7435675 0.83 MAPT (0.37) GHSRCYP2C9CYP2C19NPSR1
SCHEMBL7433678 0.81 GHSR (0.37) GHSRCYP2C9CYP2C19NPSR1
SCHEMBL7433296 0.80 CACNA1B (0.32) CTSLCACNA1BGHSRNPSR1
SCHEMBL7442699 0.80 MAPT (0.35) GHSRNPSR1
SCHEMBL7441596 0.79 GHSR (0.34) ALDH1A1GHSRNPSR1
SCHEMBL7441953 0.79 GHSR (0.35) CACNA1BGHSRRAB9A
SCHEMBL7441643 0.78 CCKAR (0.34) SLC6A4ALDH1A1GHSRNPSR1
SCHEMBL7431147 0.78 MAPT (0.40) ALDH1A1GHSRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP disclosed