SCHEMBL7443228

SCHEMBL7443228

CC(C)(C)OC(=O)CC(N)C(=O)C(C(=O)OCc1ccccc1)n1nnc(C2CCCCC2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.38
SLC6A4 P31645 1/20 0.38
CTSL P07711 1/20 0.36
CACNA1B Q00975 4/20 0.35
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
FKBP1A P62942 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SYK P43405 1/20 0.33
CAPN2 P17655 1/20 0.33
EP300 Q09472 1/20 0.33
HIF1A Q16665 1/20 0.33
CREBBP Q92793 1/20 0.33
DPP4 P27487 1/20 0.33
KCNH2 Q12809 1/20 0.33
DPP7 Q9UHL4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7436797 0.84 HTR2C (0.36) HTR2CSLC6A4CTSLCACNA1BADORA3
SCHEMBL7438701 0.82 CYP1A2 (0.48) CYP2C9CYP2C19SYK
SCHEMBL7431022 0.81 CYP1A2 (0.47) CYP2C9CYP2C19
SCHEMBL7436456 0.79 LTA4H (0.34) CTSLCACNA1BADORA3ADORA2AADORA2B
SCHEMBL7437714 0.79 CYP1A2 (0.43) CYP2C9CYP2C19
SCHEMBL7434047 0.79 CYP1A2 (0.36) CYP2C9CYP2C19SYK
SCHEMBL7443562 0.79 CYP2C9 (0.36) CYP2C9CYP2C19SYK
SCHEMBL7440427 0.78 SMN1; SMN2 (0.44) CYP2C9CYP2C19
SCHEMBL7439049 0.78 CYP1A2 (0.36) CACNA1BCYP2C9CYP2C19SYK
SCHEMBL7436644 0.77 CYP1A2 (0.35) CYP2C9CYP2C19SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP disclosed