SCHEMBL7437149

SCHEMBL7437149

CC(C)C(NC(=O)Cn1c(-c2ccccc2)ccc(N)c1=O)(O[SiH](C)C)C(C(C)(C)C)C(F)(F)C(=O)NCCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 19/20 0.50
CTRC Q99895 2/20 0.40
CMA1 P23946 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8994526 0.87 ELANE (0.58) ELANECTRC
SCHEMBL7274877 0.87 ELANE (0.56) ELANECTRC
SCHEMBL8994541 0.82 ELANE (0.51) ELANECTRC
SCHEMBL7399566 0.78 ELANE (0.62) ELANECTRCCMA1
SCHEMBL7399564 0.77 ELANE (0.53) ELANECTRCCMA1
SCHEMBL7276483 0.77 ELANE (0.59) ELANECTRC
SCHEMBL7280564 0.77 ELANE (0.61) ELANECTRC
SCHEMBL8994467 0.76 ELANE (0.55) ELANECTRCCMA1
SCHEMBL9584368 0.76 ELANE (0.51) ELANECTRCCMA1
SCHEMBL7547485 0.75 ELANE (0.75) ELANECTRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486529-A Certain pyridyl ketones for treating diseases involving leukocyte elastase ZENECA LIMITED (GB) 1996-01-23 US disclosed
EP-0636142-A1 LACTAM PEPTIDES HAVING HLE INHIBITING ACTIVITY ZENECA LIMITED (GB) 1995-02-01 EP disclosed
WO-1993021209-A1 LACTAM PEPTIDES HAVING HLE INHIBITING ACTIVITY ZENECA LIMITED (GB) 1993-10-28 WO disclosed