SCHEMBL7437241

SCHEMBL7437241

CC(C)CC(CNC(Cc1ccccc1)C(=O)CSCc1ccco1)NC(=O)OCC1CCCCCC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CTSK P43235 2/20 0.39
CTSS P25774 1/20 0.39
REN P00797 5/20 0.39
GPR88 Q9GZN0 1/20 0.38
PSMB5 P28074 3/20 0.38
PSMB1 P20618 2/20 0.38
PSMB2 P49721 2/20 0.38
POLB P06746 2/20 0.37
MMP3 P08254 1/20 0.37
USP2 O75604 1/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 1/20 0.36
BCHE P06276 1/20 0.35
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302930 0.91 PSMB1 (0.36) ALDH1A1HPGDSMN1; SMN2CTSKCTSS
SCHEMBL7305805 0.90 MGLL (0.38) ALDH1A1HPGDSMN1; SMN2
SCHEMBL7438379 0.90 CYP1A2 (0.39) ALDH1A1HPGDSMN1; SMN2PSMB5PSMB1
SCHEMBL8680990 0.89 ALDH1A1 (0.40) ALDH1A1HPGDSMN1; SMN2CTSKCTSS
SCHEMBL7437245 0.89 CAPN1 (0.46) CTSKCTSSREN
SCHEMBL7437237 0.89 CAPN1 (0.46) CTSKCTSSREN
SCHEMBL7303213 0.88 PSMB1 (0.41) ALDH1A1CTSKPSMB5PSMB1PSMB2
SCHEMBL7307063 0.88 PSMB1 (0.48) CTSKCTSSPSMB5PSMB1PSMB2
SCHEMBL7312640 0.88 PSMB1 (0.44) ALDH1A1CTSKCTSSPSMB5PSMB1
SCHEMBL7304423 0.88 PSMB1 (0.48) CTSKCTSSPSMB5PSMB1PSMB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed