SCHEMBL8680990

SCHEMBL8680990

CC(C)CC(CNC(Cc1ccccc1)C(=O)CSCc1ccco1)NC(=O)OC1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
HPGD P15428 2/20 0.40
PSMB5 P28074 3/20 0.39
PSMB1 P20618 1/20 0.39
PSMB2 P49721 1/20 0.39
POLB P06746 2/20 0.38
EDNRA P25101 2/20 0.36
TSHR P16473 4/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
LMNA P02545 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
HTT P42858 1/20 0.36
CTSL P07711 1/20 0.36
CTSS P25774 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437241 0.89 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2HPGDPSMB5PSMB1
SCHEMBL8680993 0.88 EDNRA (0.44) ALDH1A1SMN1; SMN2HPGDPSMB5PSMB1
SCHEMBL8680988 0.88 EDNRA (0.44) ALDH1A1SMN1; SMN2HPGDPSMB5PSMB1
SCHEMBL7312640 0.86 PSMB1 (0.44) ALDH1A1PSMB5PSMB1PSMB2POLB
SCHEMBL7303213 0.86 PSMB1 (0.41) ALDH1A1PSMB5PSMB1PSMB2POLB
SCHEMBL7307063 0.86 PSMB1 (0.48) PSMB5PSMB1PSMB2CTSLCTSS
SCHEMBL7304423 0.86 PSMB1 (0.48) PSMB5PSMB1PSMB2CTSLCTSS
SCHEMBL7303357 0.85 CTSS (0.46) ALDH1A1PSMB5PSMB1PSMB2POLB
SCHEMBL7436642 0.85 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2HPGDPSMB5PSMB1
SCHEMBL7305805 0.85 MGLL (0.38) ALDH1A1SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed