SCHEMBL7437601

SCHEMBL7437601

N=C(NO)c1nc(-c2ccc(OCCN3CCCCC3)cc2)cs1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 4/20 0.54
ATP4B P51164 4/20 0.54
HRH3 Q9Y5N1 3/20 0.49
ACHE P22303 2/20 0.47
LTA4H P09960 2/20 0.46
PRKAB2 O43741 1/20 0.46
PRKAG1 P54619 1/20 0.46
PRKAA2 P54646 1/20 0.46
PRKAA1 Q13131 1/20 0.46
PRKAG3 Q9UGI9 1/20 0.46
PRKAG2 Q9UGJ0 1/20 0.46
PRKAB1 Q9Y478 1/20 0.46
PRKACA P17612 1/20 0.46
ROCK1 Q13464 1/20 0.46
ESR1 P03372 2/20 0.46
ESR2 Q92731 2/20 0.46
PTPN1 P18031 1/20 0.45
PSMB1 P20618 4/20 0.44
PSMB5 P28074 4/20 0.44
PSMB2 P49721 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7440865 0.99 ATP4A (0.55) ATP4AATP4BHRH3ACHELTA4H
SCHEMBL7436848 0.83 ATP4A (0.56) ATP4AATP4BHRH3ACHELTA4H
Hydrochloric Acid SCHEMBL7438222 0.83 MCHR1 (0.52) HRH3ACHELTA4H
Hydrochloric Acid SCHEMBL7443354 0.82 ATP4A (0.57) ATP4AATP4BHRH3ACHELTA4H
SCHEMBL7437613 0.81 ATP4A (0.54) ATP4AATP4BHRH3ACHELTA4H
Hydrochloric Acid SCHEMBL7440874 0.80 ATP4A (0.55) ATP4AATP4BHRH3ACHELTA4H
SCHEMBL3612018 0.79 ACHE (0.57) ATP4AATP4BHRH3ACHELTA4H
SCHEMBL7437408 0.78 ATP4A (0.58) ATP4AATP4BHRH3LTA4HPRKAB2
Hydrochloric Acid SCHEMBL7439015 0.77 MCHR1 (0.39) ACHEPRKACAROCK1ESR1ESR2
SCHEMBL7435763 0.74 MAPT (0.55) ATP4AATP4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0506194-B1 4-aryl-thiazole or imidazole derivatives AKZO NOBEL NV (NL) 1996-08-21 EP disclosed
US-5462959-A 4-aryl-imidazole derivatives AKZO N.V. (NL) 1995-10-31 US disclosed
US-5254575-A 4-aryl-thiazole derivatives AKZO N.V. (NL) 1993-10-19 US disclosed
US-5234918-A For cardiovascular, respiratory, carcinogenic and inflammatory disorders AMERICAN CYANAMID COMPANY (US) 1993-08-10 US disclosed
EP-0506194-A1 4-aryl-thiazole or imidazole derivatives Akzo Nobel N.V. (NL) 1992-09-30 EP disclosed