SCHEMBL7439167

SCHEMBL7439167

CC(C)CC(=O)C(=O)NCC(=O)c1cccnc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 2/20 0.50
THRB P10828 1/20 0.49
PLOD3 O60568 1/20 0.46
PLOD1 Q02809 1/20 0.46
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 3/20 0.44
F7 P08709 1/20 0.44
F3 P13726 1/20 0.44
SARM1 Q6SZW1 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
SIRT6 Q8N6T7 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
SIRT3 Q9NTG7 1/20 0.44
SIRT5 Q9NXA8 1/20 0.44
SIRT4 Q9Y6E7 1/20 0.44
LMNA P02545 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC8 Q9BY41 1/20 0.43
NPC1 O15118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7436954 0.83 PLOD2 (0.53) PLOD2THRBPLOD3PLOD1KMT2A
SCHEMBL9685598 0.83 ALDH1A1 (0.52) KMT2AMEN1ALDH1A1LMNANPC1
SCHEMBL7433203 0.82 PLOD2 (0.51) PLOD2THRBPLOD3PLOD1KMT2A
SCHEMBL14073817 0.81 PLOD2 (0.59) PLOD2THRBPLOD3PLOD1KMT2A
Hydrochloric Acid SCHEMBL7441292 0.79 PLOD2 (0.48) PLOD2THRBPLOD3PLOD1KMT2A
SCHEMBL7443990 0.78 PLOD2 (0.57) PLOD2THRBPLOD3PLOD1KMT2A
SCHEMBL27374976 0.77 PLOD2 (0.49) PLOD2THRBPLOD3PLOD1ALDH1A1
SCHEMBL9565319 0.77 PLOD2 (0.46) PLOD2THRBPLOD3PLOD1KMT2A
SCHEMBL15973481 0.76 PLOD2 (0.67) PLOD2THRBPLOD3PLOD1KMT2A
SCHEMBL5113226 0.76 ALDH1A1 (0.52) PLOD2THRBPLOD3PLOD1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5278161-A Racemic mixtures HOFFMANN-LA ROCHE INC. (US) 1994-01-11 US disclosed
EP-0464572-A2 Aminoacid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-01-08 EP disclosed