SCHEMBL7439445

SCHEMBL7439445

CCC(Cc1ccccc1)c1cc(O)c(C(c2cccc(NS(=O)(=O)c3ccc(N(C)C)cc3)c2)C2CC2)c(=O)o1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK2 P53671 7/20 0.36
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
HTR6 P50406 1/20 0.35
PTGES O14684 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
LIMK1 P53667 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PGAM1 P18669 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
TGFBR1 P36897 1/20 0.33
MAP1LC3B Q9GZQ8 1/20 0.33
MAP1LC3A Q9H492 1/20 0.33
NAMPT P43490 1/20 0.33
SLC2A1 P11166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6173713 0.93 PTGES (0.38) LIMK2HTR6PTGESLIMK1ALDH1A1
SCHEMBL7444008 0.92 MAPT (0.37) LIMK2KEAP1NFE2L2HTR6ROCK2
SCHEMBL7482607 0.92 ALDH1A1 (0.40) LIMK2LIMK1ALDH1A1PGAM1MAP1LC3B
SCHEMBL6174303 0.92 ITGA1 (0.40) LIMK2PTGESLIMK1PGAM1CTSD
SCHEMBL6172890 0.91 LIMK2 (0.39) LIMK2LIMK1ALDH1A1PGAM1ADAMTS5
SCHEMBL7440371 0.91 HDAC1 (0.37) LIMK2HTR6PTGESLIMK1ALDH1A1
SCHEMBL7447436 0.91 LIMK2 (0.37) LIMK2PGAM1
SCHEMBL6175855 0.90 CYP19A1 (0.41) LIMK2KEAP1NFE2L2ALDH1A1
SCHEMBL6176577 0.90 IKBKB (0.44) KEAP1NFE2L2ALDH1A1PGAM1
SCHEMBL6174297 0.89 PGAM1 (0.38) PGAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed