SCHEMBL7440853

SCHEMBL7440853

COc1ccc2c(=O)c(N3CCNCC3)cn(Cc3ccccc3)c2c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.52
CNR2 P34972 1/20 0.52
LMNA P02545 3/20 0.48
ALDH1A1 P00352 2/20 0.48
CHRM1 P11229 1/20 0.46
TP53 P04637 1/20 0.45
PLA2G2A P14555 2/20 0.44
HTR3A P46098 2/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
MAOB P27338 1/20 0.43
HTR1A P08908 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635323 0.84 CNR1 (0.49) CNR1CNR2LMNAALDH1A1CHRM1
SCHEMBL7396359 0.82 CNR1 (0.52) CNR1CNR2LMNAALDH1A1CHRM1
SCHEMBL7017162 0.75 CHRM1 (0.62) CNR1CNR2LMNAALDH1A1CHRM1
SCHEMBL7399588 0.71 METAP1 (0.45) CNR1CNR2ALDH1A1PLA2G2A
SCHEMBL11030124 0.69 KDM4E (0.74) LMNAALDH1A1
SCHEMBL14498814 0.69 HTR3A (0.76) HTR3A
SCHEMBL7401051 0.68 DRD4 (0.42) LMNAPLA2G2A
SCHEMBL8356932 0.67 LMNA (0.73) CNR1CNR2LMNAALDH1A1CHRM1
SCHEMBL28340861 0.67 HTR6 (0.47) HTR1A
SCHEMBL4674304 0.67 HTR6 (0.71) LMNAHTR3AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5563141-A INHIBIT CELL ADHESION FOR EXAMPLE, PLATELET AGGRE GATION ZENECA LIMITED (GB) 1996-10-08 US disclosed
EP-0690847-A1 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1996-01-10 EP disclosed
WO-1994022835-A2 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1994-10-13 WO disclosed