SCHEMBL8635323

SCHEMBL8635323

COc1ccc2c(=O)c(N3CCN(c4ccncc4)CC3)cn(Cc3ccccc3)c2c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.49
CNR2 P34972 1/20 0.49
MAOB P27338 1/20 0.49
LMNA P02545 4/20 0.46
ALDH1A1 P00352 2/20 0.46
KHK P50053 2/20 0.45
CHRM1 P11229 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TP53 P04637 2/20 0.42
PLA2G2A P14555 2/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399588 0.87 METAP1 (0.45) CNR1CNR2ALDH1A1KHKPLA2G2A
SCHEMBL7401051 0.85 DRD4 (0.42) LMNAKHKPLA2G2AMAPT
SCHEMBL7440853 0.84 CNR1 (0.52) CNR1CNR2MAOBLMNAALDH1A1
SCHEMBL7396359 0.81 CNR1 (0.52) CNR1CNR2LMNAALDH1A1CHRM1
Trifluoroacetic Acid SCHEMBL8698735 0.78 SERPINE1 (0.41) CNR2LMNAMAPT
SCHEMBL5463293 0.67 CNR1 (0.43) CNR1CNR2LMNAALDH1A1CHRM1
SCHEMBL16944454 0.67 SIGMAR1 (0.60) ALDH1A1KMT2A
SCHEMBL7398283 0.66 MAPT (0.69) ALDH1A1KHKMEN1KMT2AMAPT
SCHEMBL10131759 0.65 DCTPP1 (0.40) CNR1CNR2LMNAALDH1A1MEN1
SCHEMBL8890453 0.65 GAA (0.69) LMNAALDH1A1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5563141-A INHIBIT CELL ADHESION FOR EXAMPLE, PLATELET AGGRE GATION ZENECA LIMITED (GB) 1996-10-08 US disclosed