SCHEMBL7441503

SCHEMBL7441503

N=C(N)NCc1nc(-c2ccccc2)cs1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
MAPT P10636 5/20 0.58
MEN1 O00255 4/20 0.58
LMNA P02545 4/20 0.58
KMT2A Q03164 4/20 0.58
LOXL2 Q9Y4K0 1/20 0.55
TAAR1 Q96RJ0 1/20 0.54
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
CD74 P04233 1/20 0.50
MIF P14174 1/20 0.50
MAPK1 P28482 2/20 0.47
PLAU P00749 2/20 0.47
ATP4A P20648 1/20 0.47
ATP4B P51164 1/20 0.47
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46
HDAC2 Q92769 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15125584 0.82 ALDH1A1 (0.46) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL7443407 0.81 NPC1 (0.56) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL18215350 0.79 MAPK1 (0.56) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL2227256 0.78 MAPT (0.67) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL7431740 0.78 ATP4A (0.54) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL22753445 0.77 MAPK1 (0.57) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL12890060 0.76 LOXL2 (0.58) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL22753397 0.76 MEN1 (0.55) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL9485871 0.76 HTR3A (0.65) ALDH1A1MAPTMEN1LMNAKMT2A
SCHEMBL7442912 0.74 MEN1 (0.59) ALDH1A1MAPTMEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0397364-B1 HETEROCYCLIC GUANIDINES AS 5HT 3 ANTAGONISTS PFIZER INC. (US) 1993-07-28 EP claimed
EP-0397364-A1 Heterocyclic guanidines AS 5HT 3 Antagonists PFIZER INC. (US) 1990-11-14 EP claimed
EP-0397364-B1 HETEROCYCLIC GUANIDINES AS 5HT 3 ANTAGONISTS PFIZER INC. (US) 1993-07-28 EP disclosed
US-4963689-A ANTIEMETICS, ANALGESICS, GASTROINTESTINAL DISORDERS, SCHIZOPHRENIA PFIZER INC. (US) 1990-10-16 US disclosed