SCHEMBL74422

SCHEMBL74422

CC(C)(C)OC(=O)N1CCC(Oc2ccc(OCCC(F)(F)F)cc2)CC1

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 12/20 0.60
MMP13 P45452 1/20 0.48
MMP14 P50281 1/20 0.48
CHEK2 O96017 1/20 0.47
USP30 Q70CQ3 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL75960 0.88 GPR119 (0.62) GPR119CHEK2USP30
SCHEMBL19624304 0.87 GPR119 (0.64) GPR119CHEK2
SCHEMBL23465733 0.86 GPR119 (0.62) GPR119CHEK2
SCHEMBL21023135 0.86 GPR119 (0.62) GPR119CHEK2
SCHEMBL74340 0.84 GPR119 (0.60) GPR119MMP13MMP14CHEK2
SCHEMBL6189754 0.82 GPR119 (0.64) GPR119CHEK2USP30
SCHEMBL973469 0.82 GPR119 (0.58) GPR119CHEK2
SCHEMBL19610200 0.82 GPR119 (0.58) GPR119CHEK2
SCHEMBL75039 0.82 GPR119 (0.58) GPR119MMP13MMP14CHEK2
SCHEMBL5538341 0.82 GPR119 (0.63) GPR119MMP13CHEK2USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129412-B2 Hydantoin derivatives useful as metalloproteinase inhibitors ASTRAZENECA AB (SE) 2012-03-06 US disclosed
EP-1828166-B1 HYDANTOIN DERIVATIVES USEFUL AS METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2009-07-22 EP disclosed
US-20080280950-A1 Hydantoin Derivatives Useful as Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2008-11-13 US disclosed
EP-1828166-A1 HYDANTOIN DERIVATIVES USEFUL AS METALLOPROTEINASE INHIBITORS AstraZeneca AB (SE) 2007-09-05 EP disclosed
WO-2006064218-A1 HYDANTOIN DERIVATIVES USEFUL AS METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2006-06-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080280950-A1 Hydantoin Derivatives Useful as Metalloproteinase Inhibitors MMP3, MMP9, MMP2 GPR119 2077/4885MMP13 13/4885MMP14 10/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.