SCHEMBL7444261

SCHEMBL7444261

c1ccc(Cc2cccc3[nH]c(C4CNCCN4)nc23)cc1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.57
HTR6 P50406 3/20 0.40
LTA4H P09960 1/20 0.38
HRH1 P35367 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
PARP2 Q9UGN5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1298103 0.76 PARP1 (0.80) PARP1PARP2
SCHEMBL2243349 0.74 PARP1 (0.55) PARP1HTR2B
SCHEMBL5621707 0.72 PARP1 (1.00) PARP1PARP2
Hydrochloric Acid SCHEMBL18614370 0.71 PARP1 (0.98) PARP1PARP2
SCHEMBL11380250 0.70 ALDH1A1 (0.45) HTR6LTA4H
SCHEMBL6872050 0.70 PARP1 (0.70) PARP1PARP2
SCHEMBL9307952 0.69 NPC1 (0.46) HTR6
SCHEMBL5071826 0.69 PNP (0.52)
SCHEMBL9306184 0.69 GAA (0.42) HTR6
SCHEMBL6697342 0.69 DRD2 (0.50) PARP1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628549-B1 New 1-phenylmethyl benzimidazole piperazine derivatives ESPANOLA DE PRODUCTOS FAB (ES) 2000-12-06 EP disclosed