SCHEMBL7444437

SCHEMBL7444437

N#CC1CCCC(CN(C(=O)C2(OC(=O)NCc3ccccc3)CCCCC2)C2CCNC2)C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 18/20 0.41
SLC6A4 P31645 18/20 0.41
SLC6A3 Q01959 14/20 0.41
CYP2D6 P10635 5/20 0.41
KCNH2 Q12809 4/20 0.41
CHRM4 P08173 1/20 0.39
CYP3A4 P08684 1/20 0.39
CHRM5 P08912 1/20 0.39
JAK3 P52333 1/20 0.36
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431178 0.87 JAK3 (0.38) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL6565016 0.79 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL3895614 0.77 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL3899355 0.73 HPGD (0.42)
SCHEMBL7021566 0.73 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL6565456 0.73 ACHE (0.38) JAK3OPRM1OPRD1OPRK1
SCHEMBL7431174 0.72 LMNA (0.37) JAK3OPRM1OPRD1OPRK1
SCHEMBL3898232 0.70 CTSB (0.43) OPRM1
SCHEMBL7434373 0.69 CTSB (0.40) OPRM1
SCHEMBL6564992 0.69 SLC6A4 (0.44) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed