SCHEMBL7447641

SCHEMBL7447641

CC(C)(C)ON(C=O)[C@@H](CC(F)(F)F)C(=O)C(=O)NCCCc1ccc2ccccc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.40
CES2 O00748 1/20 0.37
SIGMAR1 Q99720 3/20 0.36
CYP1A2 P05177 1/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
ASAH1 Q13510 1/20 0.34
OPRM1 P35372 1/20 0.34
SIRT5 Q9NXA8 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
VNN1 O95497 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442685 0.83 REN (0.45) RENCES2SIGMAR1CYP1A2HDAC1
SCHEMBL7443211 0.79 MMP9 (0.47) CTSK
SCHEMBL7443197 0.79 MMP9 (0.47) CTSK
SCHEMBL7442344 0.79 CTSK (0.43) MAPTHTTCTSKSMN1; SMN2
SCHEMBL7444369 0.78 EPHX1 (0.32) CTSK
SCHEMBL7444363 0.78 EPHX1 (0.32) CTSK
SCHEMBL7442591 0.78 UTS2R (0.37)
SCHEMBL7447637 0.77 CTSK (0.52) RENCES2CTSBCTSSCTSK
SCHEMBL7442741 0.77 EPHX1 (0.39)
SCHEMBL7442731 0.77 EPHX1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187905-B1 PEPTIDE COMPOUND WHICH INHIBITS VIRAL PROTEINASES; VIRICIDES FOR HEPATITIS C, HEPATITIS G, AND HUMAN GB VIRUSES HOFFMANN-LA ROCHE INC. 2001-02-13 US disclosed