SCHEMBL7447729

SCHEMBL7447729

CC(=O)Nc1cc[c]cc1OC(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
EPHX2 P34913 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
POLB P06746 2/20 0.39
KDM4E B2RXH2 1/20 0.39
RECQL P46063 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.36
BRD4 O60885 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
DYRK1A Q13627 1/20 0.36
CNR2 P34972 1/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7771748 0.81 HSD17B1 (0.46) ALDH1A1SMN1; SMN2BRD4
SCHEMBL5962103 0.78 POLB (0.56) ALDH1A1EPHX2L3MBTL1POLBKDM4E
SCHEMBL17681670 0.77 PYGL (0.48) ALDH1A1EPHX2L3MBTL1POLBKDM4E
SCHEMBL2203640 0.76 KIF11 (0.43) L3MBTL1
SCHEMBL5831442 0.75 ALDH1A1 (0.44) ALDH1A1L3MBTL1POLBKDM4ECYP2C19
SCHEMBL21268326 0.74 EPHX2 (0.38) ALDH1A1EPHX2L3MBTL1POLBKDM4E
SCHEMBL17681651 0.74 EPHX1 (0.50) ALDH1A1EPHX2L3MBTL1POLBKDM4E
SCHEMBL7399776 0.74 HDAC1 (0.46) ALDH1A1L3MBTL1POLBKDM4ECYP2C19
SCHEMBL17681776 0.73 ALDH1A1 (0.48) ALDH1A1EPHX2L3MBTL1RECQLCYP1A2
SCHEMBL17681667 0.73 CNR2 (0.62) ALDH1A1KDM4ERECQLCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043263-A (2,3-dihydrobenzofuranyl)-thiazoles as phosphodiesterase inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-03-28 US disclosed
WO-1998008844-A1 THIAZOLE DERIVATIVES USEFUL AS SELECTIVE INHIBITORS OF PDE-IV BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-03-05 WO disclosed