SCHEMBL7447763

SCHEMBL7447763

c1ccc(CCCNCc2nccs2)cc1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.53
HPGD P15428 1/20 0.51
BCHE P06276 2/20 0.48
MPO P05164 1/20 0.48
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
PLA2G4A P47712 1/20 0.46
KDM1A O60341 1/20 0.45
MAOB P27338 1/20 0.45
CES1 P23141 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7992107 0.82 KDM1A (0.50) BCHEKDM1AMAOB
SCHEMBL3223404 0.79 CES1 (0.57) SIGMAR1HPGDPLA2G4ACES1
SCHEMBL6657646 0.77 PDPK1 (0.48) PLA2G4AKDM1AMAOBCES1
SCHEMBL18956515 0.76 HTT (0.57) HPGDPLA2G4ACES1
SCHEMBL18956313 0.75 PLA2G4A (0.59) HPGDPLA2G4ACES1
SCHEMBL4730269 0.75 CYP2C19 (0.43) DRD4KDM1AMAOB
SCHEMBL29886718 0.75 HPGD (0.58) SIGMAR1HPGDPLA2G4ACES1
SCHEMBL1843939 0.74 ADRB2 (0.39) DRD4KDM1AMAOB
SCHEMBL4065566 0.74 SIGMAR1 (0.88) SIGMAR1BCHEMPO
SCHEMBL2311217 0.74 CYP2C19 (0.46) KDM1AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1200440-A1 QUINUCLIDINE DERIVATIVES FOR TREATMENT OF NEUROLOGICAL DISORDERS Vertex Pharmaceuticals Incorporated (US) 2002-05-02 EP disclosed
WO-2001002405-A1 QUINUCLIDINE DERIVATIVES FOR TREATMENT OF NEUROLOGICAL DISORDERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2001-01-11 WO disclosed