SCHEMBL7448403

SCHEMBL7448403

CN(C)C(=O)C(=O)c1c[nH]c2ccc(OCc3ccccc3)cc12

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 3/20 0.57
TRPM8 Q7Z2W7 3/20 0.57
ALDH1A1 P00352 1/20 0.56
HPGD P15428 1/20 0.56
MDH2 P40926 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
SLC6A4 P31645 1/20 0.55
LTA4H P09960 4/20 0.54
PLA2G2A P14555 4/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
HSP90AA1 P07900 1/20 0.54
HSP90AB1 P08238 1/20 0.54
KDM4E B2RXH2 1/20 0.52
MAPT P10636 1/20 0.52
KIF20A O95235 1/20 0.52
POLB P06746 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11602121 0.87 ALDH1A1 (0.61) HTR1DTRPM8ALDH1A1HPGDMDH2
SCHEMBL6098744 0.85 ALDH1A1 (0.57) HTR1DTRPM8ALDH1A1HPGDMDH2
SCHEMBL11194622 0.85 ALDH1A1 (0.59) HTR1DTRPM8ALDH1A1HPGDMDH2
SCHEMBL6764594 0.84 MAOB (0.61) HTR1DTRPM8ALDH1A1HPGDMDH2
SCHEMBL11620503 0.83 TRPM8 (0.61) HTR1DTRPM8ALDH1A1HPGDMDH2
SCHEMBL28123392 0.82 TRPM8 (0.60) HTR1DTRPM8ALDH1A1HPGDMDH2
SCHEMBL8551129 0.82 HTT (0.63) HTR1DALDH1A1MEN1KMT2AKDM4E
SCHEMBL9023222 0.82 NR4A2 (0.66) HTR1DTRPM8ALDH1A1HPGDMDH2
SCHEMBL18549394 0.82 LTA4H (0.63) HTR1DTRPM8ALDH1A1HPGDMDH2
SCHEMBL5114492 0.81 POLB (0.59) HTR1DTRPM8ALDH1A1HPGDMDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187805-B1 TREATING CONDITION FOR WHICH SELECTIVE AGONISM OR ANTAGONISM OF 5-HT-6 RECEPTORS IS INDICATED BY ADMINISTERING COMPOUNDS SUCH AS N,N-DIMETHYL 2-(1-(BENZENESULPHONYL)-5-METHOXY-1H-INDOL-3-YL)ETHYLAMINE MERCK SHARP & DOHME LTD. (GB) 2001-02-13 US disclosed