SCHEMBL7448688

SCHEMBL7448688

CC(C)[C@@H](C(=O)N[C@@H](Cc1ccc(F)cc1)C(=O)O)N(C)S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.48
ITGA4 P13612 5/20 0.48
CA2 P00918 2/20 0.44
MME P08473 6/20 0.43
ACE P12821 5/20 0.42
CPA1 P15085 4/20 0.42
ACE2 Q9BYF1 4/20 0.42
ALDH1A1 P00352 1/20 0.40
ADAMTS4 O75173 1/20 0.40
ITGB7 P26010 2/20 0.40
ECE1 P42892 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447944 0.86 MME (0.52) ITGB1ITGA4CA2MMEACE
SCHEMBL7442952 0.78 ITGB1 (0.53) ITGB1ITGA4CA2ACEALDH1A1
SCHEMBL7447863 0.77 MME (0.51) CA2MMEACECPA1ACE2
SCHEMBL7448892 0.76 MMP2 (0.53) ITGB1ITGA4CA2ACEALDH1A1
SCHEMBL7444227 0.76 ITGB1 (0.55) ITGB1ITGA4CA2ALDH1A1ADAMTS4
SCHEMBL7453817 0.75 ITGB1 (0.49) ITGB1ITGA4CA2ACEALDH1A1
SCHEMBL7448284 0.75 ITGB1 (0.49) ITGB1ITGA4CA2MMEACE
SCHEMBL7453591 0.75 MEN1 (0.52) ITGB1ITGA4CA2MMEACE
SCHEMBL7971237 0.74 ADAMTS4 (0.58) ITGB1ITGA4CA2ALDH1A1ADAMTS4
SCHEMBL7452231 0.74 MME (0.50) CA2MMEACECPA1ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221888-B1 ANTIHISTAMINE, ANTIINFLAMMATORY AGENT, AUTOIMMUNE DISEASE, RHEUMATIC DISORDERS MERCK & CO., INC. 2001-04-24 US claimed
EP-0998282-A4 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2000-08-30 EP claimed
EP-0998282-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-10 EP claimed
WO-1998053818-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed