SCHEMBL7449181

SCHEMBL7449181

C=C(C)C[C@H](NC(=O)c1ccccc1-c1csc(Nc2ccncc2)n1)C(=O)N(C)C#N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 1/20 0.39
NAMPT P43490 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
HPGDS O60760 1/20 0.36
NPC1 O15118 5/20 0.36
RAB9A P51151 5/20 0.36
MAPT P10636 3/20 0.36
GAA P10253 2/20 0.36
TP53 P04637 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MPL P40238 1/20 0.36
ALDH1A1 P00352 1/20 0.35
VCP P55072 3/20 0.35
ROCK1 Q13464 2/20 0.35
CSNK2A1 P68400 1/20 0.35
AMY1A P0DUB6 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
CASP3 P42574 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6181728 0.85 ALOX5 (0.43) NAMPTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL7449186 0.74 GRM1 (0.35) NAMPTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL7486512 0.73 CTSB (0.50) NAMPTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL7490691 0.72 CTSB (0.51) NAMPTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL6184068 0.72 CTSL (0.49) NAMPTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL6270008 0.71 SMN1; SMN2 (0.57) NAMPTSMN1; SMN2HPGDSNPC1RAB9A
SCHEMBL6181726 0.71 CTSL (0.56) NAMPTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL6265313 0.67 CTSK (0.41) NAMPTSMN1; SMN2HPGDSVCPROCK1
Trifluoroacetic Acid SCHEMBL6186180 0.66 MPL (0.39) NAMPTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL6447376 0.66 ITGB1 (0.48) CAPN1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002539192-A 2002-11-19 JP claimed
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP claimed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO claimed