SCHEMBL7449645

SCHEMBL7449645

COC(=O)[C@H](Cc1ccc(NC(=O)c2cc(NC(=N)N)cc(C(F)(F)F)c2)cc1)NC(=O)OCC(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.40
ITGAV P06756 3/20 0.40
ITGB1 P05556 3/20 0.40
ITGA2B P08514 2/20 0.40
ITGB5 P18084 2/20 0.40
ALDH1A1 P00352 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NOS3 P29474 2/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
CLPP Q16740 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
LNPEP Q9UIQ6 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458234 0.93 ITGB1 (0.47) ITGB3ITGAVITGB1ITGA2BITGB5
SCHEMBL7378843 0.93 ITGB1 (0.47) ITGB3ITGAVITGB1ITGA2BITGB5
SCHEMBL7375077 0.87 RHOC (0.39) ITGB3ITGAVNOS3NOS1NOS2
SCHEMBL7451733 0.81 FPR2 (0.45) ITGB3ITGAVITGB1ITGA2BITGB5
SCHEMBL7454545 0.81 FPR2 (0.45) ITGB3ITGAVITGB1ITGA2BITGB5
SCHEMBL7378850 0.80 ITGB1 (0.46) ITGB3ITGAVITGB1ITGA2BITGB5
SCHEMBL7458333 0.80 ITGB1 (0.46) ITGB3ITGAVITGB1ITGA2BITGB5
SCHEMBL241017 0.78 ITGB3 (0.59) ITGB3ITGAVITGB1ITGA2BITGB5
SCHEMBL241018 0.78 ITGB3 (0.59) ITGB3ITGAVITGB1ITGA2BITGB5
SCHEMBL7377736 0.78 ITGB1 (0.49) ITGB3ITGAVITGB1ITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-B1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2002-02-06 EP claimed