SCHEMBL7375077

SCHEMBL7375077

CC(C)COC(=O)N[C@@H](Cc1ccccc1)C(=O)ONC(=O)c1cc(NC(=N)N)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RHOC P08134 1/20 0.39
RHOA P61586 1/20 0.39
CTSL P07711 3/20 0.39
CTSK P43235 2/20 0.39
ITGB3 P05106 1/20 0.39
ITGAV P06756 1/20 0.39
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
FPR2 P25090 1/20 0.38
PSMB5 P28074 2/20 0.37
P2RX1 P51575 1/20 0.37
MCL1 Q07820 1/20 0.37
P2RX7 Q99572 1/20 0.36
F2 P00734 2/20 0.36
PRSS1 P07477 2/20 0.36
PRSS2 P07478 2/20 0.36
PRSS3 P35030 2/20 0.36
TACR1 P25103 2/20 0.36
TRPA1 O75762 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8428868 0.90 RHOC (0.43) RHOCRHOANOS3NOS1NOS2
SCHEMBL7458234 0.87 ITGB1 (0.47) ITGB3ITGAVFPR2P2RX1
SCHEMBL7449645 0.87 ITGB3 (0.40) RHOCRHOAITGB3ITGAVNOS3
SCHEMBL7378843 0.87 ITGB1 (0.47) ITGB3ITGAVFPR2P2RX1
SCHEMBL7380932 0.86 RHOC (0.43) RHOCRHOACTSLNOS3NOS1
SCHEMBL7382271 0.86 ITGB3 (0.48) CTSLITGB3ITGAVF2PRSS1
SCHEMBL7379710 0.80 ITGB3 (0.41) RHOCRHOACTSLITGB3ITGAV
SCHEMBL7375612 0.79 TRPA1 (0.38) RHOCRHOAFPR2P2RX1TACR1
SCHEMBL7375074 0.79 TRPA1 (0.38) RHOCRHOAFPR2P2RX1TACR1
SCHEMBL7451739 0.77 ACE (0.45) RHOCRHOAFPR2PSMB5P2RX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed