SCHEMBL7449747

SCHEMBL7449747

S=C1CSc2cc(Cl)ccc2N1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
MAOA P21397 3/20 0.40
MAOB P27338 3/20 0.40
CHRM1 P11229 3/20 0.40
PKM P14618 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAPT P10636 3/20 0.40
NOX1 Q9Y5S8 2/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
ALOX12 P18054 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
EPHX2 P34913 1/20 0.39
ALOX15 P16050 2/20 0.37
TSHR P16473 2/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
PSMB8 P28062 1/20 0.37
HAVCR2 Q8TDQ0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451860 0.87 ALDH1A1 (0.58) ALDH1A1MAOACHRM1PKMHTT
SCHEMBL7450900 0.78 ALDH1A1 (0.59) ALDH1A1MAOAMAOBMAPTNOX1
SCHEMBL4219649 0.78 MAOB (0.64) MAOAMAOBHTTMAPTSMN1; SMN2
SCHEMBL5097968 0.75 AHR (0.46) ALDH1A1CHRM1PKMHTTNPSR1
SCHEMBL88687 0.75 ALDH1A1 (1.00) ALDH1A1MAOAHTTNPSR1MAPT
SCHEMBL7450795 0.71 ALDH1A1 (0.47) ALDH1A1CHRM1
SCHEMBL8115442 0.71 SNCA (0.54) ALDH1A1CHRM1MAPTNOX1
SCHEMBL30697368 0.71 NOX1 (0.62) ALDH1A1MAOAHTTNPSR1MAPT
SCHEMBL7673182 0.71 NOX1 (0.62) ALDH1A1MAOAHTTNPSR1MAPT
SCHEMBL7448295 0.70 ALDH1A1 (0.42) ALDH1A1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed
EP-0162776-A2 Heterocyclic derivatives, process for their preparation and medicaments useful as aldose reductase inhibitors containing them LABORATOIRES UPSA (FR) 1985-11-27 EP disclosed
US-4223136-A 2,3-Dihydro-3-oxo-5H-pyrido[3,4-b][1,4]-benzothiazine-4-carbonitriles G. D. SEARLE & CO. (US) 1980-09-16 US disclosed